{"id":3994,"date":"2026-06-11T16:19:49","date_gmt":"2026-06-11T14:19:49","guid":{"rendered":"http:\/\/www.isidorolab.com\/public\/?p=3994"},"modified":"2026-06-11T16:19:54","modified_gmt":"2026-06-11T14:19:54","slug":"decoding-lysophosphatidic-acid-signaling-in-physiology-and-disease-mapping-the-multimodal-and-multinodal-signaling-networks","status":"publish","type":"post","link":"http:\/\/www.isidorolab.com\/public\/index.php\/2026\/06\/11\/decoding-lysophosphatidic-acid-signaling-in-physiology-and-disease-mapping-the-multimodal-and-multinodal-signaling-networks\/","title":{"rendered":"Decoding lysophosphatidic acid signaling in physiology and disease: mapping the multimodal and multinodal signaling networks"},"content":{"rendered":"\n<p><a href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/?term=Nadhan+R&amp;cauthor_id=41068071\">Revathy Nadhan<\/a><sup>&nbsp;<a href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/41068071\/#full-view-affiliation-1\">1<\/a><\/sup>,&nbsp;<a href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/?term=Nath+K&amp;cauthor_id=41068071\">Karthik Nath<\/a><sup>&nbsp;<a href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/41068071\/#full-view-affiliation-2\">2<\/a><\/sup>,&nbsp;<a href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/?term=Basu+S&amp;cauthor_id=41068071\">Sneha Basu<\/a><sup>&nbsp;<a href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/41068071\/#full-view-affiliation-1\">1<\/a>&nbsp;<a href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/41068071\/#full-view-affiliation-3\">3<\/a><\/sup>,&nbsp;<a href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/?term=Isidoro+C&amp;cauthor_id=41068071\">Ciro Isidoro<\/a><sup>&nbsp;<a href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/41068071\/#full-view-affiliation-4\">4<\/a><\/sup>,&nbsp;<a href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/?term=Song+YS&amp;cauthor_id=41068071\">Yong Sang Song<\/a><sup>&nbsp;<a href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/41068071\/#full-view-affiliation-5\">5<\/a><\/sup>,&nbsp;<a href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/?term=Dhanasekaran+DN&amp;cauthor_id=41068071\">Danny N Dhanasekaran<\/a><sup>&nbsp;<a href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/41068071\/#full-view-affiliation-6\">6<\/a>&nbsp;<a href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/41068071\/#full-view-affiliation-7\">7<\/a>&nbsp;<a href=\"https:\/\/pubmed.ncbi.nlm.nih.gov\/41068071\/#full-view-affiliation-8\">8<\/a><\/sup><\/p>\n\n\n\n<ul id=\"full-view-identifiers\" class=\"wp-block-list\">\n<li>PMID:\u00a0<strong>41068071<\/strong><\/li>\n\n\n\n<li>PMCID:\u00a0<a href=\"https:\/\/pmc.ncbi.nlm.nih.gov\/articles\/PMC12511386\/\" target=\"_blank\" rel=\"noreferrer noopener\">PMC12511386<\/a><\/li>\n\n\n\n<li>DOI:\u00a0<a href=\"https:\/\/doi.org\/10.1038\/s41392-025-02423-4\" target=\"_blank\" rel=\"noreferrer noopener\">10.1038\/s41392-025-02423-4<\/a><\/li>\n<\/ul>\n\n\n\n<h2 class=\"wp-block-heading\">Abstract<\/h2>\n\n\n\n<p>Lysophosphatidic acid (LPA) signaling has emerged as a central regulatory axis in both normal physiology and disease, orchestrating diverse cellular processes such as proliferation, survival, migration, immune modulation, and tissue remodeling. Originally identified as a bioactive lipid that regulates smooth muscle contraction and vascular tone, LPA has since emerged as a pleiotropic signaling molecule implicated in multiple physiological systems and a wide spectrum of pathological states. These include cancer, neurodegenerative disorders, cardiovascular and metabolic syndromes, inflammatory conditions, and fibrotic diseases. Elevated LPA levels, overexpression of autotaxin (ATX), and aberrant activation of LPA receptors (LPARs) contribute to disease initiation and progression, positioning the LPA axis as both a diagnostic biomarker and a promising therapeutic target. This review describes the multimodal and multinodal organization of the LPA signaling network, detailing upstream biosynthesis, receptor diversity, and downstream effectors across diverse organ systems. Therapeutic strategies targeting ATX, LPARs, and intracellular mediators are critically assessed, along with a review of ongoing and emerging clinical trials. Furthermore, we introduce a context-aware AI-based neural network model to simulate LPA signaling dynamics, providing a framework for predictive modeling and personalized therapeutic interventions. By integrating mechanistic insights with adaptive computational frameworks, this review positions the LPA axis as a powerful and versatile target for systems biology-guided precision medicine strategies in both health and disease.<\/p>\n\n\n\n<div data-wp-interactive=\"core\/file\" class=\"wp-block-file\"><object data-wp-bind--hidden=\"!state.hasPdfPreview\" hidden class=\"wp-block-file__embed\" data=\"http:\/\/www.isidorolab.com\/public\/wp-content\/uploads\/2026\/06\/41392_2025_Article_2423.pdf\" type=\"application\/pdf\" style=\"width:100%;height:600px\" aria-label=\"Incorporamento di 41392_2025_Article_2423.\"><\/object><a id=\"wp-block-file--media-eec6bee8-8167-4bdd-9082-3d6e75e0cc05\" href=\"http:\/\/www.isidorolab.com\/public\/wp-content\/uploads\/2026\/06\/41392_2025_Article_2423.pdf\">41392_2025_Article_2423<\/a><a href=\"http:\/\/www.isidorolab.com\/public\/wp-content\/uploads\/2026\/06\/41392_2025_Article_2423.pdf\" class=\"wp-block-file__button wp-element-button\" download aria-describedby=\"wp-block-file--media-eec6bee8-8167-4bdd-9082-3d6e75e0cc05\">Download<\/a><\/div>\n<div style='text-align:center' class='yasr-auto-insert-visitor'><!--Yasr Visitor Votes Shortcode--><div id='yasr_visitor_votes_a37f0b5f1a662' class='yasr-visitor-votes'><div class=\"yasr-custom-text-vv-before yasr-custom-text-vv-before-3994\">Clicca per votare questo articolo!<\/div><div id='yasr-vv-second-row-container-a37f0b5f1a662'\r\n                                        class='yasr-vv-second-row-container'><div id='yasr-visitor-votes-rater-a37f0b5f1a662'\r\n                                      class='yasr-rater-stars-vv'\r\n                                      data-rater-postid='3994'\r\n                                      data-rating='0'\r\n                                      data-rater-starsize='32'\r\n                                      data-rater-readonly='false'\r\n                                      data-rater-nonce='cdb0cb0a28'\r\n                                      data-issingular='false'\r\n                                    ><\/div><div class=\"yasr-vv-stats-text-container\" id=\"yasr-vv-stats-text-container-a37f0b5f1a662\"><svg xmlns=\"https:\/\/www.w3.org\/2000\/svg\" width=\"20\" height=\"20\"\r\n                                   class=\"yasr-dashicons-visitor-stats\"\r\n                                   data-postid=\"3994\"\r\n                                   id=\"yasr-stats-dashicon-a37f0b5f1a662\">\r\n                                   <path d=\"M18 18v-16h-4v16h4zM12 18v-11h-4v11h4zM6 18v-8h-4v8h4z\"><\/path>\r\n                               <\/svg><span id=\"yasr-vv-text-container-a37f0b5f1a662\" class=\"yasr-vv-text-container\">[Total: <span id=\"yasr-vv-votes-number-container-a37f0b5f1a662\">0<\/span>  Average: <span id=\"yasr-vv-average-container-a37f0b5f1a662\">0<\/span>]<\/span><\/div><div id='yasr-vv-loader-a37f0b5f1a662' class='yasr-vv-container-loader'><\/div><\/div><div id='yasr-vv-bottom-container-a37f0b5f1a662' class='yasr-vv-bottom-container'><\/div><\/div><!--End Yasr Visitor Votes Shortcode--><\/div>","protected":false},"excerpt":{"rendered":"<p>Revathy Nadhan&nbsp;1,&nbsp;Karthik Nath&nbsp;2,&nbsp;Sneha Basu&nbsp;1&nbsp;3,&nbsp;Ciro Isidoro&nbsp;4,&nbsp;Yong Sang Song&nbsp;5,&nbsp;Danny N Dhanasekaran&nbsp;6&nbsp;7&nbsp;8 Abstract Lysophosphatidic acid (LPA) signaling has emerged as a central regulatory axis in both normal physiology and disease, orchestrating diverse cellular processes such as proliferation, survival, migration, immune modulation, and tissue remodeling. Originally identified as a bioactive lipid that regulates smooth muscle contraction and vascular tone,&hellip;<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"closed","ping_status":"closed","sticky":false,"template":"","format":"standard","meta":{"yasr_overall_rating":0,"yasr_post_is_review":"","yasr_auto_insert_disabled":"","yasr_review_type":"","footnotes":""},"categories":[1],"tags":[],"class_list":["post-3994","post","type-post","status-publish","format-standard","hentry","category-senza-categoria"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v26.8 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\r\n<title>Decoding lysophosphatidic acid signaling in physiology and disease: mapping the multimodal and multinodal signaling networks - IsidoroLab<\/title>\r\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\r\n<link rel=\"canonical\" href=\"http:\/\/www.isidorolab.com\/public\/index.php\/2026\/06\/11\/decoding-lysophosphatidic-acid-signaling-in-physiology-and-disease-mapping-the-multimodal-and-multinodal-signaling-networks\/\" \/>\r\n<meta property=\"og:locale\" content=\"it_IT\" \/>\r\n<meta property=\"og:type\" content=\"article\" \/>\r\n<meta property=\"og:title\" content=\"Decoding lysophosphatidic acid signaling in physiology and disease: mapping the multimodal and multinodal signaling networks - IsidoroLab\" \/>\r\n<meta property=\"og:description\" content=\"Revathy Nadhan&nbsp;1,&nbsp;Karthik Nath&nbsp;2,&nbsp;Sneha Basu&nbsp;1&nbsp;3,&nbsp;Ciro Isidoro&nbsp;4,&nbsp;Yong Sang Song&nbsp;5,&nbsp;Danny N Dhanasekaran&nbsp;6&nbsp;7&nbsp;8 Abstract Lysophosphatidic acid (LPA) signaling has emerged as a central regulatory axis in both normal physiology and disease, orchestrating diverse cellular processes such as proliferation, survival, migration, immune modulation, and tissue remodeling. 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